Local anesthetics

Local anesthetics reduce or completely suppress the excitability of sensory nerve endings in the mucous membranes, skin and other tissues in direct contact. Depending on the method of application of local anesthetic distinguish between terminal anesthesia (anesthetic is applied to the surface, where it blocks the end of the sensitive nerves), infiltration (the anesthetic solution is consistently "impregnate" the skin and deeper tissues), conduction (the anesthetic is injected along the nerve, causing the block of conduction of excitation along the nerve fibers), spinal anesthesia (subarachnoid anesthetic is administered).

The first substance that has discovered exhibits activity, was the alkaloid cocaine. Due to the high toxicity it is currently almost not used. In modern anesthesiology is the use of a number of synthetic local anesthetics. These include procaine, trimekain, tetracaine (mainly in ophthalmology), lidocaine. Recently with long-established local anesthetics (bupivacaine, etc.).

The scope of different drugs depending on their pharmacological and physico-chemical properties: benzocaine as an insoluble substance applies only superficially. Soluble drugs are used for different types of local anesthesia.

Some local anesthetics possess anti-arrhythmic activity. Lidocaine has a relatively wide application in certain types of arrhythmias. For the same purpose is used trimekain.



Acriol Pro (Lidocaine + Prilocaine) 2.5% + 2.5% cream

Acriol Pro (Lidocaine + Prilocaine) 2.5% + 2.5% cream

Expiration date: 06/2019 INN: lidocaine + prilocaine Pharmacotherapeutic group: local anes..

$7.98

Anaesthesol 10 suppositories

Anaesthesol 10 suppositories

Expiration date: 05/2020 The composition and form of issue: Suppositories for rectal appli..

$4.87

Aurobin 20g ointment

Aurobin 20g ointment

Expiration date: 03/2019 The composition and form of issue:Ointment 1 tube contains:prednisolon..

$9.74

Benoxi (Oxybuprocaine) 10mg/ml 10ml eye drops

Benoxi (Oxybuprocaine) 10mg/ml 10ml eye drops

Expiration date: 09/2018 Composition1 ml vial containing 4 mg oxybuprocaine hydrochloridePackag..

$6.04

BloccoC (Bupivacaine) 5mg/ml 4ml 5 vials

BloccoC (Bupivacaine) 5mg/ml 4ml 5 vials

Expiration date: 11/2020 In may 2011 the Russian pharmaceutical market, new drug BloccoC p..

$30.76

Bupivacaine 5mg/ml 4ml 5 vials

Bupivacaine 5mg/ml 4ml 5 vials

Expiration date: 08/2019 Action: Local anesthetic Composition:Bupivacaine - 5mgIndica..

$15.58

Cathejell (Lidocaine + Chlorhexidine) gel

Cathejell (Lidocaine + Chlorhexidine) gel

Expiration date: 12/2021 The composition and form of issue: 100 g of gel for topical use c..

$6.81

Dentinox 10g gel

Dentinox 10g gel

Expiration date: 03/2021 The composition and form of issue: 1 year dental solution or gel ..

$13.63

Emla (Lidocaine + Prilocaine) cream

Emla (Lidocaine + Prilocaine) cream

Expiration date: 08/2019 The composition and form of issue: Cream for local and external u..

$56.46

Inokain (Oxybuprocaine) 0.4% 5ml eye drops

Inokain (Oxybuprocaine) 0.4% 5ml eye drops

Expiration date: 06/2019 Structure and Composition:Drops eye 0.4%. 1 ml contains:oxybuproc..

$4.87

Kamistad (Lidocaine + Chamomillae recutitae floridis extract) 10g gel

Kamistad (Lidocaine + Chamomillae recutitae floridis extract) 10g gel

Expiration date: 11/2021 The composition and form of issue: Gel for local application. 100..

$9.74

Lidocaine

Lidocaine

Expiration dates: %2 vials 09/2020, 10% vials 11/2019 CompositionIn 1 liter of solution for inj..

$3.89

Lidocaine 10% spray 50ml

Lidocaine 10% spray 50ml

Expiration date: 08/2019 Action: topical anesthetic Composition: lidocaine hydro..

$15.58

Lidocaine 10% spray 50ml

Lidocaine 10% spray 50ml

Expiration date: 03/2020 Structure and Composition:1g metered spray contains 3.8 g of lidocaine..

$23.36

Marcaine Spinal (Bupivacaine) 0.5% 4ml 5 vials

Marcaine Spinal (Bupivacaine) 0.5% 4ml 5 vials

Expiration date: 10/2018 Structure and Composition: Injection. 1 ml contains: bupivac..

$23.36

Marcaine Spinal Heavy (Bupivacaine) 0.5% 4ml 5 vials

Marcaine Spinal Heavy (Bupivacaine) 0.5% 4ml 5 vials

Expiration date: 02/2019 CompositionActive substance: bupivacaine hydrochloride monohydrate for..

$36.51

Menovasin (Benzocaine + Procaine + Racementhol) 40ml solution

Menovasin (Benzocaine + Procaine + Racementhol) 40ml solution

Expiration date: 09/2019 The composition and form of issue: 100 ml solution of 70% ethyl a..

$2.34

Menovasin (Benzocaine + Procaine + Racementhol) 50ml solution

Menovasin (Benzocaine + Procaine + Racementhol) 50ml solution

Expiration date: 11/2020 Action: local anesthetic Composition: L-menthol, n..

$4.09

Novocaine (Procaine)

Novocaine (Procaine)

Expiration date: 03/2020  Structure and Composition Novocaine - injection:1 ml s..

$3.60

Novocaine (Procaine) 100mg 10 suppositories

Novocaine (Procaine) 100mg 10 suppositories

Expiration date: 09/2018 Pharmachologic effect: Local anesthetic activity with moderate an..

$2.73

Otipax 15ml drops

Otipax 15ml drops

Expiration date: 03/2022 The composition and form of issue: 100 g ear drops contain p..

$8.57

Otirelax (Lidocaine + Phenazone) 15ml ear drops

Otirelax (Lidocaine + Phenazone) 15ml ear drops

Expiration date: 07/2020 The composition and form of issue: Ear drops. 1 g contains:active..

$7.79

Procto-Glyvenol (Tribenoside + Lidocaine)

Procto-Glyvenol (Tribenoside + Lidocaine)

Expiration date: 04/2022 The composition and form of issue: 1 rectal suppository contains ..

$11.68

Relief Advance (Benzocaine)

Relief Advance (Benzocaine)

Expiration date: 01/2019 Structure and Composition: Ointment for rectal and external appli..

$9.74

Ropivacaine

Ropivacaine

Expiration date: 03/2020 Excipients: sodium chloride - 7.59 mg hydrochloric acid q.s.to pH..

$38.94

Ultracain D-S (Articaine)

Ultracain D-S (Articaine)

Expiration date: 06/2020 Structure and Composition: 1 ml injection solution contains ..

$37.97

Ultracain D-S forte (Articaine)

Ultracain D-S forte (Articaine)

Expiration date: 06/2020 Structure and Composition: 1 ml injection solution contains 40 mg..

$37.97

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